Rhizome of Chinese Goldthread — Safety & Interactions

Chuan Huang Lian · Rhizoma Coptidis

Contraindications

  • Spleen and Stomach deficiency cold — primary TCM contraindication
  • Yin deficiency with secondary Heat signs
  • Blood deficiency patterns with secondary Heat
  • Jaundiced neonates — berberine displaces bilirubin; do not administer to newborns with jaundice

Cautions

  • May prolong QTc interval in patients with underlying heart disease; use with caution in cardiac conditions
  • Use with caution during pregnancy — intensely cold properties may disturb gestational balance
  • Breastfeeding: use with caution; berberine transfers into breast milk

Drug Interactions

Drug Class / Substrate Mechanism Severity Source
CYP2D6, CYP2C9, and CYP3A4 substrate drugs Huanglian inhibits CYP2D6, CYP2C9, and CYP3A4; may increase plasma levels and side effects of substrate drugs. Prolonged use may also induce CYP3A4, potentially decreasing drug concentrations Unknown Memorial Sloan Kettering

This information is for educational purposes only and does not constitute medical advice. Always consult a qualified healthcare provider before using herbal medicines, especially if you take prescription medications.