Use with caution. Review interactions and contraindications below.
TCM Properties
- Taste
- bitter
- Temperature
- cold
- Channels
- Lung, Gallbladder, Spleen, Large Intestine, Small Intestine, Heart, Stomach
Traditional Use
Primary Actions
- Clears Heat and dries Dampness
- Purges Fire and resolves toxicity
- Stops bleeding due to Blood Heat
- Calms the fetus
Secondary Actions
- Drains Heat from the upper burner
- Clears Lung Heat and stops cough
Classic Formulas
- Xiao Chai Hu Tang — addresses half-exterior, half-interior conditions with alternating fever and chills
- Huang Qin Tang — treats Heat-driven diarrhea with abdominal pain
Classical References
- Shang Han Lun (Zhang Zhongjing): Huang Qin is the principal herb for clearing Heat from the Shaoyang interior
Modern Research
Active Compounds
- Baicalein
- Baicalin
- Wogonin
- Wogonoside
- Oroxylin A
Studied Effects
- Baicalein induces apoptosis in non-small cell lung cancer by inhibiting the glutamine-mTOR metabolic pathway (PMID 38432394)
- Baicalein triggers ferroptosis in colorectal cancer cells via JAK2/STAT3/GPX4 axis suppression (PMID 38684798)
- Total flavonoids exhibit cardiovascular protective effects via multiple mechanisms (PMID 36152591)
PubMed References
Safety & Interactions
Contraindications
- Spleen-Stomach deficiency cold
- Cold-type diarrhea
- Lung cold with cough
- Blood deficiency conditions
- Kidney Yang deficiency with loose stools
Cautions
- Hepatotoxicity reported in case reports; monitor liver function with prolonged use
- Pneumonitis (lung inflammation) reported rarely
- May elevate triglycerides and high-sensitivity C-reactive protein
Drug Interactions
-
Anticoagulants and antiplatelets (e.g., warfarin)
— Baicalin has antithrombotic activity; additive effect may increase bleeding risk (Moderate)
Source: Memorial Sloan Kettering
-
Statins (HMG-CoA reductase inhibitors)
— Decreases blood levels of statin drugs, reducing cholesterol-lowering efficacy; documented in healthy volunteers (Moderate)
Source: Memorial Sloan Kettering
-
CYP1A2 and CYP2C19 substrates
— Wogonin inhibits CYP1A2 and CYP2C19 enzymes; may increase plasma levels and adverse effects of affected drugs (Unknown)
Source: Memorial Sloan Kettering
-
SLC transporter substrates
— Baicalein, baicalin, and wogonin inhibit SLC uptake transporters; may alter pharmacokinetics of co-administered drugs (Unknown)
Source: Memorial Sloan Kettering